Rational Design of Macrocyclic Noncovalent Inhibitors of SARS-CoV-2 Mpro from a DNA-Encoded Chemical Library Screening Hit That Demonstrate Potent Inhibition Against Pan-Coronavirus Homologues and Nirmatrelvir-Resistant Variants. Xu Wang,Dimitar Gotchev,Kristi Yi Fan, Marvin M. Vega,Nagraj Mani, Kayleigh McGovern-Gooch,Andrea Cuconati, Breanna Tercero,Xiaohe Wang, Philip Carpino,Klaus Maskos,Paolo A. Centrella, Andreas Schmitt, Franziska Preuss, Archna Prasad, Chia-yi Chen,Matthew A. Clark,John P. Guilinger, Shawn Johnstone, Konstanze von Konig,Anthony D. Keefe, Jenny Liu, Stephane Turcotte,Ying Zhang, Debora L. Konz Makino,Angela M. Lam,Andrew G. Cole,Michael J. SofiaJOURNAL OF MEDICINAL CHEMISTRY(2024)引用 0|浏览2AI 理解论文溯源树样例生成溯源树,研究论文发展脉络Chat Paper正在生成论文摘要