BBO-8520, a First-in-class, Direct Inhibitor of KRASG12C (ON), Locks GTP-bound KRASG12C in the State 1 Conformation Resulting in Rapid and Complete Blockade of Effector BindingAnna E. Maciag, James Stice, Bin Wang,Alok Sharma,Albert Chan, Ken Lin, Devansh Singh,Marcin Dyba,Yue Yang, Saman Setoodeh, Brian P. Smith,Dana Rabara, Zuhui Zhang,Erik K. Larsen, Dom Esposito,John Paul Denson,Michela Ranieri,Mary Meynardie,Sadaf Mehdizadeh,Patrick Alexander,Maria Abreu Blanco,David Turner,Rui Xu,Felice C. Lightstone,Kwok Kin Wong,Dhirendra Simanshu,Keshi Wang,Andrew G. Stephen,Kerstin Sinkevicius,Dwight V. Nissley,Eli Wallace,Frank McCormick,Pedro J. BeltranCANCER RESEARCH(2024)引用 0|浏览10AI 理解论文溯源树样例生成溯源树,研究论文发展脉络Chat Paper正在生成论文摘要