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Exploring Structure-Activity Relationships of Pyrrolyl Diketo Acid Derivatives As Non-Nucleoside Inhibitors of Terminal Deoxynucleotidyl Transferase Enzyme.

Valentina Noemi Madia, Nadia Garibaldi,Davide Ialongo, Elisa Patacchini, Valeria Tudino, Giuseppe Ruggieri, Laura Zarbo, Emanuele Cara,Antonio Coluccia, Marco Artico,Luigi Scipione,Antonella Messore,Francesco Saccoliti, Elisa Mentegari,Giovanni Maga,Roberto Di Santo,Emmanuele Crespan,Roberta Costi

Journal of enzyme inhibition and medicinal chemistry(2025)

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Key words
DNA repair,terminal deoxynucleotidyl transferase,medicinal chemistry,drug discovery,structure–activity relationships
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