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Crystallographic Fragment Screening and Deep Mutational Scanning of Zika Virus NS2B-NS3 Protease Enable Development of Resistance-Resilient Inhibitors.

Frank von Delft,Xiaomin Ni, R Richardson,Andre Godoy, Matteo Ferla,Caroline Kikawa,Jenke Scheen, William Hannon, Eda Capkin, Noa Lahav, Blake Balcomb,Peter Marples,Michael Fairhead,SiYi Wang, Eleanor Williams,Charles Tomlinson, Jasmin Aschenbrenner, Ryan Lithgo,Max Winokan,Charline Giroud, Anu Chandran,Martin Walsh,Warren Thompson,Jesse Bloom,Haim Barr,Karla Kirkegaard,Lizbé Koekemoer,Daren Fearon, Matthew Evans

Research square(2025)

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