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Discovery of Non-Covalent Inhibitors for SARS-CoV-2 PLpro: Integrating Virtual Screening, Synthesis, and Experimental Validation

Bruna K. P. Sousa,Melina Mottin, Donald Seanego, Christopher D. Jurisch, Beatriz S. A. Rodrigues, Veronica L. S. da Silva,Milene Aparecida Andrade, Gilberto S. Morais Jr, Diogo F. Boerin, Thamires Q. Froes,Flavia Nader Motta,M. Cristina Nonato,Izabela D. M. Bastos,Kelly Chibale,Richard K. Gessner,Carolina Horta Andrade

ACS MEDICINAL CHEMISTRY LETTERS(2024)

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关键词
SARS-CoV-2,COVID-19,papain-like protease(PLpro),virtual screening,synthesis,enzymatic assay,noncovalent inhibitor,naphthyridine
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