Development of a Series of Pyrrolopyridone MAT2A Inhibitors
Stephen J. Atkinson,Sharan K. Bagal,Argyrides Argyrou,Sean Askin,Tony Cheung,Elisabetta Chiarparin,Muireann Coen,Iain T. Collie,Ian L. Dale,Claudia De Fusco,Keith Dillman,Laura Evans,Lyman J. Feron,Alison J. Foster,Michael Grondine,Vasudev Kantae,Gillian M. Lamont,Scott Lamont,James T. Lynch,Sten Nilsson Lill,Graeme R. Robb,Jamal Saeh,Marianne Schimpl,James S. Scott,James Smith,Bharath Srinivasan,Sharon Tentarelli,Mercedes Vazquez-Chantada,David Wagner,Jarrod J. Walsh,David Watson,Beth Williamson Journal of Medicinal Chemistry(2024)
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Transition State Analogue Inhibitors
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