Rational Optimization of a Transcription Factor Activation Domain Inhibitor
Shaon Basu,Paula Martínez-Cristóbal,Marta Frigolé-Vivas,Mireia Pesarrodona,Michael Lewis,Elzbieta Szulc,C. Adriana Bañuelos,Carolina Sánchez-Zarzalejo,Stasė Bielskutė,Jiaqi Zhu,Karina Pombo-García,Carla Garcia-Cabau, Levente Zodi, Hannes Dockx,Jordann Smak, Harpreet Kaur,Cristina Batlle,Borja Mateos,Mateusz Biesaga,Albert Escobedo,Lídia Bardia,Xavier Verdaguer,Alessandro Ruffoni,Nasrin R. Mawji,Jun Wang,Jon K. Obst,Teresa Tam,Isabelle Brun-Heath,Salvador Ventura,David Meierhofer,Jesús García,Paul Robustelli,Travis H. Stracker,Marianne D. Sadar,Antoni Riera,Denes Hnisz,Xavier Salvatella Nature Structural & Molecular Biology(2023)
Key words
Transcription Factors,Transcriptional Regulation,Drug Discovery Paradigm
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