Identification of an Orally Bioavailable, Brain-Penetrant Compound with Selectivity for the Cannabinoid Type 2 Receptor.
Molecules(2022)
关键词
cannabinoid receptors CB1,CB2,pyrrolobenzodiazepines,neuroinflammation,neurodegenerative diseases,central nervous system (CNS),pharmacokinetics (PK),radioligand binding assay
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