Discovery Of Bms-812204, A Cannabinoid Receptor (Cb1) Antagonist, Via Reductions In Log P In The Series To Balance Volume Of Distribution And Clearance Bruce A. Ellsworth , Ximao Wu , Philip M. Sher , Gang Wu , Amarendra Mikkilineni , Zhengxiang Gu , Natesan Murugesan , Yeheng Zhu , Guixue Yu , Doree Sitkoff , Kenneth Carlson , Liya Kang , Yifan Yang , Ning Lee , Roseann Baska , Qi Huang , William Keim , Mary Jane Cullen , Eva Zuvich , Michael Thomas , Kenneth W. Rohrbach , James J. Devenny , Helen Godonis , Susan Harvey , Brian J. Murphy , Gerry Everloff , Paul Stetsko , Olafur Gudmundsson , Susan Johnghar , Asoka Ranasinghe , Kamelia Behnia , Maryann Pelleymounter , William R. Ewing ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY(2009)
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