Design, Synthesis and Biological Evaluation of 2-H Pyrazole Derivatives Containing Morpholine Moieties As Highly Potent Small Molecule Inhibitors of APC–Asef Interaction
European journal of medicinal chemistry(2019)
关键词
APC,Asef,Colorectal cancer,Small-molecule inhibitors,Docking simulation,Orthotopic transplantation model
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