Design, Synthesis and Biological Evaluation of Indane Derived GPR40 Agopams.
Barbara Pio,Harry R. Chobanian,Yan Guo,Hubert Josien,William K. Hagmann,Michael Miller,Maria E. Trujillo,Melissa Kirkland,Daniel Kosinski,Joel Mane,Michele Pachanski,Boonlert Cheewatrakoolpong,Eric Ashley,Robert Orr,Michael J. Wright,Randal Bugianesi,Sarah Souza,Xiaoping Zhang,Jerry Di Salvo,Adam B. Weinglass,Richard Tschirret-Guth,Koppara Samuel,Qing Chen,Jackie Shang,James Lamca,Juliann Ehrhart,Ravi Nargund,Andrew D. Howard,Steven L. Colletti Bioorganic & Medicinal Chemistry Letters(2019)
Key words
GPR40 AgoPAM,FFA1,GPCR,Diabetes,Indane
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