Discovery of Chromane Propionic Acid Analogues As Selective Agonists of GPR120 with in Vivo Activity in Rodents.
Gregory L. Adams,Francisco Velazquez,Charles Jayne,Unmesh Shah,Shouwu Miao,Eric R. Ashley,Maria Madeira,Taro E. Akiyama,Jerry Di Salvo,Takao Suzuki,Nengxue Wang,Quang Truong,Eric Gilbert,Dan Zhou,Andreas Verras,Melissa Kirkland,Michele Pachanski,Maryann Powles,Wu Yin,Feroze Ujjainwalla,Srikanth Venkatraman,Scott D. Edmondson ACS Medicinal Chemistry Letters(2016)
关键词
GPR120,FFAR4,insulin sensitization,type 2 diabetes,chromane
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