Discovery of 7-Aminofuro[2,3-c]pyridine Inhibitors of Tak1: Optimization of Kinase Selectivity and Pharmacokinetics
Keith R. Hornberger,Dan M. Berger,Andrew P. Crew,Hanqing Dong,Andrew Kleinberg,An-Hu Li,Matthew R. Medeiros,Mark J. Mulvihill,Kam Siu,James Tarrant,Jing Wang,Felix Weng,Victoria L. Wilde,Mark Albertella,Mark Bittner,Andrew Cooke,Michael J. Gray,Paul Maresca,Earl May,Peter Meyn, William Peick,Darlene Romashko,Michael Tanowitz,Brianna Tokar Bioorganic & Medicinal Chemistry Letters(2013)
关键词
TAK1,Inhibitors,7-Amino-furo[2,3-c]pyridine,Cancer,Inflammation
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